Pyrazino (1,2-a) - and 1,4-diazepino (1,2-a) indoles. II. Synthesis of 1-substituted 10-phenyl-3,4-dihydropyrazino (1,2-a) indoles and of 11-phenyl-4,5-dihydro-4H-diazepino (1,2-a) indoles
Gatta, F.; Zaccari, V.; Huidobro-Toro, J.P.; Chiavarelli, S.
Il Farmaco; Edizione Scientifica 30(1): 58-69
1975
ISSN/ISBN: 0430-0920 PMID: 1116593 Document Number: 86388
The AA. describe the synthesis of some 1-substituted 10-phenyl-3,4-dihydropyrazino(1,2-a)indoles and 11-phenyl-4,5-dihydro-3H-1,4-diazepino(1,2-a)indoles. Preliminary pharmacological tests indicate that these products, have lower sedative and antiadrenergic activity than the compounds reported in our previous paper.
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