Top Abstract Purchase Related
Home
>
Node
>
Subnode

Synthesis, characterization and antimicrobial evaluation of some new 1,3-thiazole-2,4-diamine derivatives

Siddiqui, N.; Shaquiquzzaman; ur Rahman, M.; Arshad, M.F.; Ahsan, W.; Alam, M.S.; Ahmed, S.

Acta Poloniae Pharmaceutica 67(3): 239-246

2010

ISSN/ISBN: 0001-6837
PMID: 20524425
Document Number: 641855
Various N,N'-diaryl-1,3-thiazole-2,4-diamines (3a-w) were synthesized by a three steps process. The structures of the synthesized compounds were confirmed by spectral data and elemental analyses. All the synthesized compounds were tested against two bacterial strains and two fungal strains. Bacterial strains included Gram positive Staphylococcus aureus and Gram negativeve Escherichia coli and fungal strains included Monascus purpurea and Penicillium citrinum. Most of the compounds showed moderate to good antibacterial as well as antifungal activity.

Document emailed within 1 workday
Secure & encrypted payments

Kharchenko, S.N.; Litvin, V.P.; Pis' ko, G.T. 1978: Antimicrobial properties of hexamethylene diamine and piperidine derivatives Mikrobiolohichnyi Zhurnal 40(1): 76-79
Raffa, D.; Migliara, O.; Daidone, G.; Maggio, B.; Schillaci, D. 2002: Synthesis and antimicrobial evaluation of new phenoxyacetamide derivatives Bollettino Chimico Farmaceutico 141(1): 3-7
Kosáry, J.; Kasztreiner, E.; Rablóczky, G.; Vitális, B. 1987: Synthesis of thiazole derivatives with positive inotropic effect Die Pharmazie 42(6): 373-375
Kotb, E.R.; Soliman, H.A.; Morsy, E.M.H.; Abdelwahed, N.A.M. 2017: New Pyridine and Triazolopyridine Derivatives: Synthesis, Antimicrobial and Antioxidant Evaluation Acta Poloniae Pharmaceutica 74(3): 861-872
Geronikaki, A.; Sotiropoulou, E.; Kourounakis, P. 1989: Synthesis of some thiazole derivatives with prospective local anaesthetic activity Die Pharmazie 44(5): 349
Deep, A.; Kumar, P.; Narasimhan, B.; Lim, S.M.; Ramasamy, K.; Mishra, R.K.; Mani, V. 2016: Synthesis, Antimicrobial, Anticancer Evaluation and Qsar Studies of Thiazolidin-4-One Derivatives Acta Poloniae Pharmaceutica 73(1): 93-106
Adeel-Sharif, H.M.; Ahmed, D.; Mir, H. 2015: Antimicrobial salicylaldehyde Schiff bases: synthesis, characterization and evaluation Pakistan Journal of Pharmaceutical Sciences 28(2): 449-455
Zawadzka, J.; Bogdal, M. 1984: Thiazole derivatives. V. Synthesis and pharmacological screening of amides of 4-phenyl-5-thiazolecarboxylic acids Acta Poloniae Pharmaceutica 41(6): 633-640
Rüttinger, H.H.; Dehne, H.; Schroth, W. 1976: Reactivity and biological effect in the thiazole series. 1. a new synthesis of thiazole with the N-acylthioamides Die Pharmazie 31(4): 218-221
Mohsen, A.; Omar, M.E.; Salama, H.M.; Eshba, N.H. 1985: Novel thiazolidine-2,4-dione-4-thiosemicarbazone and 4-[(3,4-diaryl-3H-thiazol-2-yl)azo]thiazolidin-2-one derivatives: synthesis and evaluation for antimicrobial and anticancer properties Il Farmaco; Edizione Scientifica 40(1): 49-57
Aftab, K.; Aslam, K.; Kousar, S.; Nadeem, M.J.U.H. 2016: Synthesis, characterization and biological evaluation of tryptamine based benzamide derivatives Pakistan Journal of Pharmaceutical Sciences 29(2): 423-428
Aboul-Enein, M.N.; El-Difrawy, S.M.; Nofal, Z.M.; El-Azzouny, A.A.; El-Hawary, S. 1982: Synthesis and antimicrobial activity of 2-arylmethylpyrrolidine derivatives Acta Pharmaceutica Suecica 19(4): 309-316
Basoglu, S.; Yolal, M.; Demirci, S.; Demirbas, N.; Bektas, H.; Karaoglu, S.A. 2013: Design, synthesis and antimicrobial activities of some azole derivatives Acta Poloniae Pharmaceutica 70(2): 229-236
Patel, P.; Koregaokar, S.; Shah, M.; Parekh, H. 1996: Synthesis of some novel pyrazoline and cyanopyridine derivatives as antimicrobial agents Farmaco 51(1): 59-63
Hassan, E.; Al-Ashmawi, M.I.; Abd El-Fattah, B. 1983: Synthesis and antimicrobial testing of certain oxadiazoline and triazole derivatives Die Pharmazie 38(12): 833-835
Habib, N.S.; Abdel-Hamid, S.; el-Hawash, M. 1989: Synthesis of benzimidazole derivatives as potential antimicrobial agents Farmaco 44(12): 1225-1232
Chawla, R.; Arora, A.; Parameswaran, M.K.; Chan, P.; Sharma, D.; Michael, S.; Ravi, T.K. 2010: Synthesis of novel 1,3,4-oxadiazole derivatives as potential antimicrobial agents Acta Poloniae Pharmaceutica 67(3): 247-253
el-Naggar, A.M.; Hussein, M.E.; el-Nemma, E.M.; Samour, A.A. 1985: Synthesis and antimicrobial activity of some new isonicotinoylamino acid and dipeptide derivatives Il Farmaco; Edizione Scientifica 40(9): 662-670
Kozminykh, V.O.; Igidov, N.M.; Kozminykh, E.N.; Semenova, Z.N.; Andreichikov YuS 1992: Synthesis and antimicrobial activity of new 5-aryl-2-hydroxy-3(2H)-pyrrolinone derivatives Die Pharmazie 47(4): 261-263
el-Shaaer, H.M.; Abdel-Aziz, S.A.; Allimony, H.A.; Ali, U.F.; Abdel-Rahman, R.M. 1997: Synthesis and antimicrobial activities of some new 2-substituted benzoxazole/benzothiazole derivatives Die Pharmazie 52(8): 585-589