1,2,3-triazole derivatives of arylalkanoic acids
Da Settimo, A.; Livi, O.; Ferrarini, P.L.; Tonetti, I.; Ciabattini, E.
Il Farmaco; Edizione Scientifica 34(5): 371-382
1979
ISSN/ISBN: 0430-0920 PMID: 554790 Document Number: 139360
A series of several 1,2,3-triazole derivatives, by reaction of p-azidophenylacetic and 2-(p-azidophenyl)propionic acids with active methylene compounds, was synthesized. Some of the derivatives obtained were subjected to pharmacological study and among these compounds (II m) showed an analgesic activity 2.5 times greater than phenylbutazone.
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