Preliminary screening of anticholinergic effect of some new derivatives of glycolic and aminoacetic acids
Faff, J.; Woliński, J.; Bandolet, J.; Bak, W.
Polish Journal of Pharmacology and Pharmacy 30(4): 497-499
1978
ISSN/ISBN: 0301-0244 PMID: 740551 Document Number: 125649
The anticholinergic effect of some new alkylaminoalkyl esters of benzilic, cyclohexyl, 1-hydroxycyclohexyl, piperidino-and morpholino acetic acids (Table 1) was evaluated. Only benzilic acid esters were active and the 2-N-piperidinoaminoethyl benzilate hydrochloride (ANC-30) has the highest pA2 value.
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