Synthesis and biological activity of new analogs of beta-casomorphine-5
Sobirov, M.M.; Khalikov, S.Kh.; Saidov, S.S.; Kodirov, M.Z.; Zaĭtsev, S.V.; Chichenkov, O.N.; Varfolomeev, S.D.
Bioorganicheskaia Khimiia 20(7): 740-750
1994
ISSN/ISBN: 0132-3423 PMID: 7993378 Document Number: 428301
The level of affinity and the degree of selectivity of the peptides towards the mu- and delta-opioid receptors of the rat brain lyophilized membranes were studied by the radioreceptor method. All the new peptides displayed analgetic activity, largely depending upon their structure.
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