Synthesis of 3-phenyl-3-phenylthiopropionic acids, amides, amines and studies on their pharmacological properties
Mirek, J.; Chojnacka-Wójcik, E.; Tatarzyńska, E.; Wiczyńska, B.
Il Farmaco; Edizione Scientifica 40(9): 701-708
1985
ISSN/ISBN: 0430-0920 PMID: 4076432 Document Number: 265208
The addition of mercaptobenzene to cinnamic acids yielded 3-phenyl-3-phenylthiopropionic acids which were then converted to the amides. The latter compounds were reduced to the amines with lithium aluminum hydride. Some of the obtained amides displayed significant biological activity.
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