Potential long-acting contraceptive agents: esters and ethers of testosterone with alpha- and/or beta-chain branching
Herz, J.E.; Torres, J.V.; Murillo, A.; Cruz, S.; Shafiee, A.; Vosooghi, M.; Sotheeswaran, S.; Gunatilaka, A.A.
Steroids 46(6): 947-953
1985
ISSN/ISBN: 0039-128X PMID: 3842023 DOI: 10.1016/s0039-128x(85)80002-7Document Number: 424595
The synthesis of ten esters and two ethers of testosterone (17 beta-hydroxyandrost-4-en-3-one) is described. All these possess some form of alpha - and/or beta - substitution in the ester/ether side-chain. The work was undertaken in order to evaluate the long-acting antifertility effect of such compounds in males.
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