Methyl N- (diphenylmethyl) -D,L-tryptophanates: synthesis and benzodiazepine receptor affinity
Balsamini, C.; Duranti, E.; Salvatori, A.; Spadoni, G.; Barone, D.
Farmaco 45(10): 1111-1117
1990
ISSN/ISBN: 0014-827X PMID: 1965622 Document Number: 353507
Several Methyl N-(diphenylmethyl)-D,L-tryptophanates were synthetized and the affinity for the central benzodiazepine receptor was measured. Disappointingly, none of the tested compounds showed to be active, even at the high concentration examined.
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