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Synthesis and in vitro antimicrobial study of 4-thiazolidinone containing sulfanilamide

Zevzikoviene, A.; Zevzikovas, A.; Tarasevicius, E.; Pavlonis, A.; Dirse, V.

Acta Poloniae Pharmaceutica 69(5): 911-915

2012

ISSN/ISBN: 0001-6837
PMID: 23061287
Document Number: 658167
The title compounds, 3-allyl-2-sulfanylamido-4-thiazolidinones (2a-d), have been synthesized after substitution of amino group of sulfanylamide with allylisothiocyanate and cyclization into 4-thiazolidinones. The synthesized compounds were tested for their antibacterial and antifungal activity (MIC) in vitro) against microorganisms: S. aureus, E. faecalis. E. coli, P. aeruginosa, K. pneumoniae, P. mirabilis, B. subtilis, B. cereus and C. albicans taking sulfadimidine, sulfathiazole, sulfanilamide and sulfamethizole as standard drugs. Synthesized compounds (2a-d) demonstrated selective activity against B. cereus.

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