Short peptides containing L-lysine and epsilon-aminocaproic acid as potential plasmin inhibitors
Purwin, M.; Bruzgo, I.; Markowska, A.; Midura-Nowaczek, K.
Die Pharmazie 64(11): 765-767
2009
ISSN/ISBN: 0031-7144 PMID: 20099524 Document Number: 632264
Eight short peptides containing L-lysine and epsilon-aminocaproic acid were obtained and their effect on the amidolytic activities of plasmin, thrombin and trypsin was examined. Tripeptide amide Boc-EACA-L-Lys-EACA-NH2 was the most effective and specific plasmin inhibitor.
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