Synthesis and antibacterial activity of eremomycin esters through the carboxyl group
Pavlov, A.I.; Olsuf'eva, E.N.; Berdnikova, T.F.; Rozynov, B.V.; Aleksandrova, L.G.; Malkova, I.V.; Preobrazhenskaia, M.N.
Bioorganicheskaia Khimiia 17(6): 849-854
1991
ISSN/ISBN: 0132-3423 PMID: 1776969 Document Number: 377828
Methyl, benzyl and diphenylmethyl esters of the glycopeptide antibiotic eremomycin were obtained by its treatment with corresponding diazoalkanes. The esters have high antibacterial activity but are less active than the parent antibiotic.
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