Reversal of multidrug resistance by non-antitumor anthracycline analogs

Inaba, M.; Nagashima, K.; Sakurai, Y.; Fukui, M.; Yanagi, Y.

Gan 75(12): 1049-1052

1984


ISSN/ISBN: 0016-450X
PMID: 6597118
Document Number: 232967
It was found that three synthetic anthracycline analogs lacking not only antitumor activity but also calcium-antagonizing action possessed an activity to potentiate vincristine cytotoxicity against vincristine-resistant P388 leukemia. ID-8279, one of these analogs, significantly reversed resistance to vincristine and daunorubicin by increasing their intracellular accumulation.

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