Syntheses of new 5,6,7,8-tetrahydropyrrolo [2,3-d]azepine ring system
Waly, M.A.
Bollettino Chimico Farmaceutico 139(5): 217-221
2000
ISSN/ISBN: 0006-6648 PMID: 11213441 Document Number: 514153
A first synthesis of pyrrolo[2,3-d]azepine ring system starting from pyrrole and perhydroazepine derivatives was reported. In addition, Lansbury's reaction is developed through the use of para-toluene sulphonic acid (p-TsOH) as a new catalyst for this reaction.
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